4,6-二氟-2,3-二氢吲哚合成路线 (共 1 条)
反应条件
triethylsilane; trifluoroacetic acid in dichloromethane T=0 - 20°C; 4 h;
参考文献
PFIZER INC.; Bhattacharya, Samit; Cameron, Kimberly; Dowling, Matthew; Fernando, Dilinie; Ebner, David; Filipski, Kevin; Kung, Daniel; Lee, Esther; Smith, Aaron; Tu, Meihua
Patent: US2013/267493 A1, 2013 ;
Location in patent: Paragraph 0719 ;