反应条件
1: With formic acid; triethylamine in DMF (N,N-dimethyl-formamide) T=95°C; 2 h; 2: With hydrogenchloride; water in DMF (N,N-dimethyl-formamide) pH=1;
参考文献
Griebenow, Nils; Flessner, Timo; Buchmueller, Anja; Raabe, Martin; Bischoff, Hilmar; Kolkhof, Peter
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 8 p. 2554 - 2558