2-[4-(溴甲基)苯基]-1,1,1,3,3,3-六氟丙烷-2-醇合成路线 (共 2 条)
反应条件
N-bromosuccinmide; 2,2'-azo-bisisobutyronitrile in tetrachloromethane T=20°C; 50 h; Heating / reflux;
参考文献
PHARMACIA CORPORATION
Patent: WO2003/99775 A1, 2003 ;
Location in patent: Page 16 ;
反应条件
N-bromosuccinmide; 2,2'-azo-bisisobutyronitrile in tetrachloromethane T=80°C; 2 h;
参考文献
WO2013/166013 A1, ;
Paragraph 0085 ;