反应条件
1: SOCl2 / CHCl3 / 4 h / 65 °C 2: Na2CO3, Et3N / methanol / 1 h / 65 °C 3: 1.) n-BuLi, LiC10H7 / 1.) THF, hexane, -78 deg C, 3 h, 2.) THF, hexane, from -78 to 20 deg C, overnight View Scheme
参考文献
Tetrahedron Asymmetry, , vol. 7, # 10 p. 2911 - 2922