反应条件
1: in N,N-dimethyl-formamide T=13 - 17°C; 3 h; Large scale; 2: in N,N-dimethyl-formamide T=75 - 80°C; 1 h; Large scale;
参考文献
Conlon, David A.; Drahus-Paone, Antoinette; Ho, Guo-Jie; Pipik, Brenda; Helmy, Roy; McNamara, James M.; Shi, Yao-Jun; Williams, J. Michael; Macdonald, Dwight; Deschenes, Denis; Gallant, Michel; Mastracchio, Anthony; Roy, Bruno; Scheigetz, John
Organic Process Research and Development, 2006 , vol. 10, # 1 p. 36 - 45