反应条件
1: toluene / -78 °C 2: 62 percent / PhSH, BF3*Et2O / CH2Cl2 / 0 °C 3: 96 percent / 2,6-lutidine / CH2Cl2 / 0 °C 4: Pd2(dba)3PPh3-Et3N / toluene / 6 h / 120 °C 5: camphorsulfonic acid / methanol View Scheme
参考文献
Konno, Katsuhiro; Maki, Shojiro; Fujishima, Toshie; Zhaopeng, Liu; Miura, Daishiro; Chokki, Manabu; Takayama, Hiroaki
Bioorganic and Medicinal Chemistry Letters, 1998 , vol. 8, # 2 p. 151 - 156