反应条件
1: 300 mg / Na2S2O4 / methanol; H2O / Ambient temperature 2: 252 mg / CH2Cl2 / Ambient temperature 3: 258 mg / NaI / acetone / 4 h / Heating 4: i-Pr2NEt / acetonitrile / 80 °C 5: H2, Et3N / Pd/C / ethanol; tetrahydrofuran / 1 h / 760 Torr View Scheme
参考文献
Hamill, Terence G.; Brenner, Nancy J.; Eng, Wai-Si; Burns, H. Donald
Journal of Labelled Compounds and Radiopharmaceuticals, 1998 , vol. 41, # 4 p. 319 - 327