反应条件
1: 55 percent / 1 N NaOH / methanol / 1.5 h / 25 °C 2: 40 percent / H3PO4, DMSO, N,N'-dicyclohexylcarbodiimide / 1.5 h / 25 °C View Scheme
参考文献
Iqbal, Nadeem; Akula, Murthy R.; Vo, Dean; Matowe, Wandikayi C.; McEwen, Carol-Anne; Wolowyk, Michael W.; Knaus, Edward E.
Journal of Medicinal Chemistry, 1998 , vol. 41, # 11 p. 1827 - 1837