1-[(2S,3S,4S,5S)-3,4-二羟基-5-(羟基甲基)四氢呋喃-2-基]-1,2,4-三唑-3-甲酰胺合成路线 (共 1 条)
反应条件
With methanol; ammonia T=20°C; Hydrolysis; amination; 18 h;
参考文献
Ramasamy, Kanda S.; Tam, Robert C.; Bard, Josie; Averett, Devron R. Journal of Medicinal Chemistry, 2000 , vol. 43, # 5 p. 1019 - 1028