2-溴丙二醛合成路线

参考文献

Hartmann, Rolf; Frotscher, Martin; Oberwinkler, Sandrine; Ziegler, Erika; Messinger, Josef; Thole, Heinrich-Hubert
Patent: US2010/204234 A1, 2010 ;
Location in patent: Page/Page column 12 ;
US 20100204234 A1

2065-75-02-溴丙二醛+

1225387-53-0

705263-10-16-溴-吡唑[1,5-a]咪唑+

875781-17-25-溴-1H-吡唑并[3,4-b]吡啶

参考文献

WO2006/128692 A2, ;

Page/Page column 86 ;

2065-75-02-溴丙二醛+

1225387-53-0

875781-17-25-溴-1H-吡唑并[3,4-b]吡啶

参考文献

ARRAY BIOPHARMA INC.; GENENTECH, INC.; AHRENDT, Kateri A.; BUCKMELTER, Alexandre J.; DE MEESE, Jason; GRINA, Jonas; HANSEN, Joshua D.; LAIRD, Ellen R.; LUNGHOFER, Paul; MORENO, David; NEWHOUSE, Brad; REN, Li; SEO, Jeongbeob; TIAN, Hongqi; WENGLOWSKY, Steven Mark; FENG, Bainian; GUNZNER, Janet; MALESKY, Kim; MATHIEU, Simon; RUDOLPH, Joachim; WEN, Zhaoyang; YOUNG, Wendy B.
Patent: WO2009/111279 A1, 2009 ;
Location in patent: Page/Page column 79-80 ;
WO 2009/111279 A1

1820-80-03-氨基吡唑+

2065-75-02-溴丙二醛

875781-17-25-溴-1H-吡唑并[3,4-b]吡啶

参考文献

ELI LILLY AND COMPANY
Patent: WO2006/52568 A2, 2006 ;
Location in patent: Page/Page column 23-24 ;
WO 2006/052568 A2

1072-98-62-氨基-5-氯吡啶+

2065-75-02-溴丙二醛

29096-59-16-氯咪唑并[1,2-a]吡啶-3-甲醛

参考文献

Bioorganic and Medicinal Chemistry, , vol. 15, # 1 p. 403 - 412

2065-75-02-溴丙二醛+

352-34-1对氟碘苯

957062-56-54-溴-1-(4-氟苯基)-1H-吡唑

参考文献

Gerstenberger, Brian S.; Rauckhorst, Mark R.; Starr, Jeremy T.
Organic Letters, 2009 , vol. 11, # 10 p. 2097 - 2100

1820-80-03-氨基吡唑+

2065-75-02-溴丙二醛

705263-10-16-溴-吡唑[1,5-a]咪唑

参考文献

THE GENERAL HOSPITAL CORPORATION; THE BRIGHAM AND WOMEN'S HOSPITAL, INC.
Patent: WO2009/114180 A1, 2009 ;
Location in patent: Page/Page column 71 ;

2065-75-02-溴丙二醛+

1225387-53-0

705263-10-16-溴-吡唑[1,5-a]咪唑+

875781-17-25-溴-1H-吡唑并[3,4-b]吡啶

参考文献

WO2006/128692 A2, ;

Page/Page column 86 ;

2065-75-02-溴丙二醛+

1225387-53-0

705263-10-16-溴-吡唑[1,5-a]咪唑

参考文献

Cuny, Gregory D.; Yu, Paul B.; Laha, Joydev K.; Xing, Xuechao; Liu, Ji-Feng; Lai, Carol S.; Deng, Donna Y.; Sachidanandan, Chetana; Bloch, Kenneth D.; Peterson, Randall T.
Bioorganic and Medicinal Chemistry Letters, 2008 , vol. 18, # 15 p. 4388 - 4392

504-29-02-氨基吡啶+

2065-75-02-溴丙二醛

6188-43-8咪唑并[1,2-a]吡啶-3-甲醛

参考文献

UCB S.A.
Patent: WO2006/128692 A2, 2006 ;
Location in patent: Page/Page column 64; 65 ;