1: With sodium hydroxide in methanol T=90°C; 16 h; 2: With hydrogenchloride in methanol; water pH=Ca.3;
参考文献
THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK; SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH; BRESLOW, Ronald; MARKS, Paul, A.
Patent: WO2013/52110 A1, 2013 ;
Location in patent: Page/Page column 63; 64; 65 ;