2-氯-N,N-二甲基-4-吡啶羧酰胺合成路线 (共 1 条)
反应条件
benzotriazol-1-ol; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride; triethylamine in water; N,N-dimethyl-formamide T=20°C; 17 h;
参考文献
TAISHO PHARMACEUTICAL CO., LTD.; ARENA PHARMACEUTICALS, INC.
Patent: WO2006/35967 A1, 2006 ;
Location in patent: Page/Page column 91 ;
WO 2006/035967 A1