2-氟-4-(4-吗啉)苯胺合成路线 (共 2 条)
反应条件
1: 1.81 g / tetrahydrofuran / 2 h / 20 °C 2: 8.4 percent / H2 / Pd/C / methanol / 2.5 h / 2327.17 Torr View Scheme
参考文献
Patil, Sudhakar G.; Bagul, Rahul R.; Swami, Mangesh S.; Kotharkar, Nandini; Darade, Kalpana
Chinese Chemical Letters, 2011 , vol. 22, # 8 p. 883 - 886
反应条件
potassium carbonate; copper monobromide
参考文献
Bristol-Myers Squibb Pharma Company
Patent: EP946508 B1, 2009 ;
Location in patent: Page/Page column 94 ;