反应条件
1: 1.) BuLi, HMPT / 1.) THF, -78 deg C, 5 min, 2.) THF, RT, overnight 2: LiOH, LiBr, Bu4NBr / acetonitrile / 1 h View Scheme
参考文献
Karoyan, Philippe; Sagan, Sandrine; Clodic, Gil; Lavielle, Solange; Chassaing, Gerard
Bioorganic and Medicinal Chemistry Letters, 1998 , vol. 8, # 11 p. 1369 - 1374