反应条件
benzotriazol-1-ol; O-(1H-benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium hexafluorophosphate; N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide T=20°C;
参考文献
Barry, Grant D.; Suen, Jacky Y.; Le, Giang T.; Cotterell, Adam; Reid, Robert C.; Fairlie, David P.
Journal of Medicinal Chemistry, 2010 , vol. 53, # 20 p. 7428 - 7440