反应条件
1: 93 percent / NaIO4 / H2O; methanol / 16 h / Ambient temperature
2: 60 percent / TFAA / benzene / 151 h / Ambient temperature; other N-(aryl)methyl-2-(phenylsulfinyl)ethylamines, also with TFAA and BF3*Et2O
3: 64 percent / NaBH4, NiCl2*6H2O / methanol; tetrahydrofuran / 0.5 h / Ambient temperature
4: 89 percent / 10percent aq. NaOH / ethanol / Ambient temperature
View Scheme
参考文献
Shinohara, Tatsumi; Takeda, Akira; Toda, Jun; Ueda, Yoko; Kohno, Michiyo; Sano, Takehiro
Chemical and Pharmaceutical Bulletin, 1998 , vol. 46, # 6 p. 918 - 927
