6-(氯甲基)-N,N-二甲基-1,3,5-三嗪-2,4-二胺合成路线 (共 2 条)
反应条件
1: [99Tc]-Metformin hydrochloride With sodium methylate in methanol T=20°C; 3 h; 2: chloroacetic acid methyl ester in methanol 30 h;
参考文献
Brzozowski; Saczewski; Gdaniec
European Journal of Medicinal Chemistry, 2000 , vol. 35, # 12 p. 1053 - 1064
反应条件
sodium methylate in methanol T=20°C;
参考文献
Inamdar, Gajanan S.; Pandya, Amit N.; Thakar, Hardik M.; Sudarsanam, Vasudevan; Kachler, Sonja; Sabbadin, Davide; Moro, Stefano; Klotz, Karl-Norbert; Vasu, Kamala K.
European Journal of Medicinal Chemistry, 2013 , vol. 63, p. 924 - 934