反应条件
1: 95 percent / CH2Cl2 / 0.5 h / 0 °C 2: 1,2-dimethoxy-ethane / -15 °C 3: NaBH4 4: 1.) (COCl)2, DMSO, 2.) Et3N / 1.) CH2Cl2, -78 deg C, 15 min, 2.) CH2Cl2, -78 deg C, 5 min View Scheme
参考文献
Martin, Loic; Cornille, Fabrice; Coric, Pascale; Roques, Bernard P.; Fournie-Zaluski, Marie-Claude
Journal of Medicinal Chemistry, 1998 , vol. 41, # 18 p. 3450 - 3460
