4-(叔-丁基二甲基硅烷基)氧基-2-硝基苯胺合成路线 (共 2 条)
反应条件
1H-imidazole in dichloromethane T=20°C; Cooling with ice;
参考文献
BEIGENE, LTD.; ZHOU, Changyou; WANG, Shaohui; ZHANG, Guoliang
Patent: WO2013/97224 A1, 2013 ;
Location in patent: Page/Page column 61 ;
反应条件
in ethyl acetate; N,N-dimethyl-formamide
参考文献
Eli Lilly and Company
Patent: US6313122 B1, 2001 ;
US 6313122 B1