反应条件
1: (1-methyl-1H-[1,2,3]triazol-4-yl)methanol With lithium hexamethyldisilazane in tetrahydrofuran; N,N-dimethyl-formamide T=-10°C; 0.5 h; 2: 6-chloro-3-(5-methylisoxazol-3-yl)-1,2,4-triazolo[3,4-a]phthalazine in tetrahydrofuran; N,N-dimethyl-formamide T=20°C; 16 h;
参考文献
Sternfeld, Francine; Carling, Robert W.; Jelley, Richard A.; Ladduwahetty, Tamara; Merchant, Kevin J.; Moore, Kevin W.; Reeve, Austin J.; Street, Leslie J.; O'Connor, Desmond; Sohal, Bindi; Atack, John R.; Cook, Susan; Seabrook, Guy; Wafford, Keith; Tattersall, F. David; Collinson, Neil; Dawson, Gerard R.; Castro, Jose L.; MacLeod, Angus M.
Journal of Medicinal Chemistry, 2004 , vol. 47, # 9 p. 2176 - 2179