2-(4-吡啶)噻唑-5-羧酸合成路线 (共 1 条)
反应条件
potassium carbonate; tetrakis(triphenylphosphine) palladium(0) in 1,4-dioxane; water T=160°C; 0.333333 h; Microwave irradiation;
参考文献
Millennium Pharmaceuticals, Inc.
Patent: US2008/171754 A1, 2008 ;
Location in patent: Page/Page column 95 ;
US 20080171754 A1