去乙酰基雷奈佐利硫代乙酰胺合成路线 (共 2 条)
反应条件
Lawesson's reagent in 1,4-dioxane
T=20°C; 20.5 h; Heating / reflux;
参考文献
Pharmacia and Upjohn Company
Patent: US6342513 B1, 2002 ;
Location in patent: Page column 30-31 ;
反应条件
potassium hydroxide; NAF in ethanol
T=20°C; 8.66667 h;
参考文献
Pharmacia and Upjohn Company
Patent: US6342513 B1, 2002 ;
Location in patent: Page column 34 ;