1-N-甲磺酰基-4-哌啶酮合成路线 （共 7 条）
反应条件
sodium hydroxide in tetrahydrofuran; water T=20 - 32°C; 2 h;
参考文献
US2004/34008 A1, ;
Page/Page column 12 ;
US 20040034008 A1
反应条件
potassium carbonate in acetone
反应条件
1: With oxalic acid in tetrahydrofuran; water 1 h; Heating / reflux; 2: With acetic acid in tetrahydrofuran; water 3 h; Heating / reflux;
参考文献
EP993460 B1, ;
Page 35 ;
反应条件
triethylamine in dichloromethane T=0°C; 4 h;
参考文献
WO2006/26760 A2, ;
Page/Page column 141 ;
参考文献
WO2007/122410 A1, ;
Page/Page column 100 ;
反应条件
1: in acetonitrile T=20°C; 1 h; 2: With sodium tris(acetoxy)borohydride in acetonitrile T=-10 - 20°C; 3: With sodium hydroxide in water
参考文献
US2004/34008 A1, ;
Page/Page column 12-13 ;
US 20040034008 A1
反应条件
aq. NaOH; NaBH(OAc)3; CH3NH2 in acetonitrile
