1-(5-碘-2-吡啶基)哌嗪合成路线 (共 3 条)
反应条件
trifluoroacetic acid T=20°C; 0.5 h;
参考文献
Bioorganic and Medicinal Chemistry, , vol. 15, # 4 p. 1586 - 1605
反应条件
potassium carbonate in acetonitrile
参考文献
Resolution Pharmaceuticals, Inc.
Patent: US5976497 A1, 1999 ;
US 5976497 A
反应条件
1: 79 percent / Et3N / ethanol / 72 h / Heating 2: TFA / 0.5 h / 20 °C View Scheme
参考文献
Bioorganic and Medicinal Chemistry, , vol. 15, # 4 p. 1586 - 1605