反应条件
1: p-bromophenyl mercaptan With potassium carbonate in N,N-dimethyl-formamide T=0 - 20°C; 0.25 h; 2: 4-fluoro-nitro-benzene in N,N-dimethyl-formamide T=80°C; 16 h;
参考文献
FORMA THERAPEUTICS, INC.; GENENTECH, INC.; BAIR, Kenneth W.; BAUMEISTER, Timm B.; BUCKMELTER, Alexandre J.; CLODFELTER, Karl H.; HAN, Bingsong; LIN, Jian; REYNOLDS, Dominic J.; SMITH, Chase C.; WANG, Zhongguo; ZHENG, Xiaozhang; YUEN, Po-Wai
Patent: WO2012/31196 A1, 2012 ;
Location in patent: Page/Page column 237 ;
WO 2012/031196 A1