3-(3,4-二氯苯基)-2-丙炔-1-醇合成路线 (共 2 条)
反应条件
copper(l) iodide; triethylamine; bis-triphenylphosphine-palladium(II) chloride in tetrahydrofuran T=35°C; 12 h;
参考文献
DOV PHARMACEUTICAL, INC.
Patent: WO2008/57575 A2, 2008 ;
Location in patent: Page/Page column 60-61 ;
反应条件
Product distribution / selectivity;
参考文献
GLAXO GROUP LIMITED
Patent: WO2008/31771 A2, 2008 ;
Location in patent: Page/Page column 45-46 ;