3-氟-4-(4-甲基-1-哌嗪基)苯胺合成路线 (共 3 条)
反应条件
palladium in ethanol; ethyl acetate
参考文献
SUNSHINE LAKE PHARMA CO., LTD.; ZHANG, Yingjun; ZHANG, Jiancun; WANG, Xiaojun; LIN, Runfeng; CAO, Shengtian; WANG, Zhaohe; LI, Jing
Patent: WO2014/12360 A1, 2014 ;
Location in patent: Paragraph 00293 ;
反应条件
1: 49 percent / 100 °C 2: H2 / Pd/C / ethanol / 16 h / 20 °C View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 49, # 16 p. 4981 - 4991
反应条件
1: 49 percent / 100 °C 2: H2 / Pd/C / ethanol / 16 h / 20 °C View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 49, # 16 p. 4981 - 4991