反应条件
1: 97 percent / H2 / Pd/C 2: 77 percent / TBAF / tetrahydrofuran 3: 1.) SO2Cl2, 2.) MeOH 4: 75 percent / TFA / CH2Cl2 5: 1.) MsCl, Et3N, 2.) DBU / 2.) THF View Scheme
参考文献
Lew, Willard; Williams, Matthew A.; Mendel, Dirk B.; Escarpe, Paul A.; Kim, Choung U.
Bioorganic and Medicinal Chemistry Letters, 1997 , vol. 7, # 14 p. 1843 - 1846