反应条件
1: 5-bromo-4-chloro-7H-pyrrolo[2,3-d]pyrimidine With sodium hydride in N,N-dimethyl-formamide T=0°C; 0.5 h; 2: benzenesulfonyl chloride in N,N-dimethyl-formamide T=20°C; 2 h;
参考文献
Blake, James F.; Kallan, Nicholas C.; Xiao, Dengming; Xu, Rui; Bencsik, Josef R.; Skelton, Nicholas J.; Spencer, Keith L.; Mitchell, Ian S.; Woessner, Richard D.; Gloor, Susan L.; Risom, Tyler; Gross, Stefan D.; Martinson, Matthew; Morales, Tony H.; Vigers, Guy P.A.; Brandhuber, Barbara J.
Bioorganic and Medicinal Chemistry Letters, 2010 , vol. 20, # 19 p. 5607 - 5612