反应条件
1: triethylamine / (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride / 100 °C / 15001.5 Torr / Inert atmosphere; autoclave vessel 2: toluene-4-sulfonic acid / methanol / 2 h / 20 °C View Scheme
参考文献
PHENEX PHARMACEUTICALS AG; KREMOSER, Claus; ABEL, Ulrich; STEENECK, Christoph; KINZEL, Olaf
Patent: WO2011/20615 A1, 2011 ;
