反应条件
1: 82 percent / NaOAc / ethyl acetate; H2O / 4 h / Ambient temperature 2: 87 percent / H2 / 5percent Pd/C / acetic acid; HClO4 / 24 h / 30 °C / 2280 Torr 3: 67 percent / 25percent HCl / 1.) methanol, 90 deg C, 6 h; 2.) r.t., 17 h View Scheme
参考文献
Horn, Alan S.; Kaptein, Bernard; Vermue, Niek A.; Vries, Jan B. De; Mulder, Theo B. A.
European Journal of Medicinal Chemistry, 1988 , vol. 23, p. 325 - 328
