1: With lithium hydroxide hydrate; water in tetrahydrofuran T=20°C; 4 h; 2: With hydrogenchloride in water pH=3 - 4; Product distribution / selectivity;
参考文献
Conrig Pharma ApS; Hansen, John Bondo; Thomsen, Mikael Søndergaard
Patent: US2013/303497 A1, 2013 ;
Location in patent: Paragraph 0279-0281 ;