1: With iodine; magnesium in tetrahydrofuran Metallation; 12 h; Heating; 2: With boric acid trimethyl ester in tetrahydrofuran T=20°C; Substitution; 3: With hydrogenchloride in tetrahydrofuran T=0 - 5°C; Hydrolysis; Further stages.;
参考文献
Zhang, Fang-Jie; Cortez, Cecilia; Harvey, Ronald G.
Journal of Organic Chemistry, 2000 , vol. 65, # 13 p. 3952 - 3960