反应条件
1: NaBH4 / ethanol / 1) 0.5h, RT 2) 0.5h, reflux
2: 1) POCl3 2) Et3N / 1) CH2Cl2, 24h 2) 2h, ice cooling
View Scheme
参考文献
Modak, A. S.; Sahasrabudhe, S. D.
Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry, 1984 , vol. 23, # 10 p. 980 - 982