1: With sulfuric acid; boric acid; sodium nitrite in water T=0 - 130°C; 2: With ammonium hydroxide in water T=20°C; pH=8 - 9;
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Vernekar, Sanjeev Kumar V.; Hallaq, Hasan Y.; Clarkson, Guy; Thompson, Andrew J.; Silvestr, Linda; Lummis, Sarah C. R.; Lochner, Martin
Journal of Medicinal Chemistry, 2010 , vol. 53, # 5 p. 2324 - 2328
THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL; JIN, Jian; ROTH, Bryan; FRYE, Stephen
Patent: WO2012/3418 A2, 2012 ;
Location in patent: Page/Page column 73-74 ;
WO 2012/003418 A2
Vernekar, Sanjeev Kumar V.; Hallaq, Hasan Y.; Clarkson, Guy; Thompson, Andrew J.; Silvestr, Linda; Lummis, Sarah C. R.; Lochner, Martin
Journal of Medicinal Chemistry, 2010 , vol. 53, # 5 p. 2324 - 2328