反应条件
1: 1,2,3-Benzotriazole With sodium methylate in methanol 2: chloromethyl-trimethyl-silane With 18-crown-6 ether in N,N-dimethyl-formamide
参考文献
Roman, Bart I.; Ryck, Tine De; Dierickx, Laura; Vanhoecke, Barbara W.A.; Katritzky, Alan R.; Bracke, Marc; Stevens, Christian V.
Bioorganic and Medicinal Chemistry, 2012 , vol. 20, # 15 p. 4812 - 4819