1: With N-(diphenylmethylene)amine; 2,2'-bis-(diphenylphosphino)-1,1'- binaphthyl; sodium t-butanolate; tris(dibenzylideneacetone)dipalladium (0) in toluene 2: With hydrogenchloride in tetrahydrofuran Further stages.;
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 17, # 22 p. 6378 - 6382
hydrogen bromide; copper(I) bromide; sodium nitrite in water T=0 - 75°C; Sandmeyer reaction; 12.5 h; Inert atmosphere;
参考文献
Shi, Jun; Manolikakes, Georg; Yeh, Chien-Hung; Guerrero, Carlos A.; Shenvi, Ryan A.; Shigehisa, Hiroki; Baran, Phil S.
Journal of the American Chemical Society, 2011 , vol. 133, # 20 p. 8014 - 8027
