1: 5-[(3AS,4S,6AR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl]pentanoic acid With benzotriazol-1-ol; dicyclohexyl-carbodiimide in N,N-dimethyl-formamide 0.166667 h; 2: monopropargylamine in N,N-dimethyl-formamide T=20°C;
参考文献
Chemistry - A European Journal, , vol. 16, # 18 p. 5416 - 5424