反应条件
hydrogenchloride; phosphate buffer; sodium hydrogencarbonate 1.) 100 deg C, 80 min, 2.) CH3OH, 71 deg C, 3.5 d; Yield givenMultistep reaction;
参考文献
Bergeron, Raymond J.; Wiegand, Jan; McManis, James S.; McCosar, Bruce H.; Weimar, William R.; Brittenham, Gary M.; Smith, Richard E.
Journal of Medicinal Chemistry, 1999 , vol. 42, # 13 p. 2432 - 2440