1-氟-4-[(4-硝基苯基)磺酰基]苯合成路线 (共 4 条)
反应条件
potassium carbonate in acetonitrile T=20 - 25°C; 16 h;
参考文献
PHARMACIA and UPJOHN COMPANY
Patent: WO2004/96809 A1, 2004 ;
Location in patent: Page 16 ;
WO 2004/096809 A1
参考文献
Journal of Medicinal Chemistry, , vol. 17, # 1 p. 142 - 144
参考文献
Magnetic Resonance in Chemistry, , vol. 25, p. 1001 - 1006
反应条件
hydrazine hydrate; palladium on activated charcoal
参考文献
American Cyanamid Company
Patent: US4532349 A1, 1985 ;