反应条件
benzotriazol-1-ol; triethylamine; dicyclohexyl-carbodiimide in N,N-dimethyl-formamide 1.) 4 deg C, 48 h, 2.) RT, 3 days;
参考文献
Dutta, Anand S.; Gormley, James J.; McLachlan, Peter F.; Major, John S.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 9 p. 2552 - 2560