triethylamine in 1,4-dioxane; dichloromethane
T=0 - 20°C; 16 h;
参考文献
Radyukhin, V. A.; Kazakova, N. A.; Filippovich, E. I.; Evstigneeva, R. P.
J. Gen. Chem. USSR (Engl. Transl.), 1982 , vol. 52, # 2 p. 432 - 440,377 - 384
sodium hydrogencarbonate in tetrahydrofuran; water
16 h; Ambient temperature;
参考文献
Chu, Daniel T. W.; Nordeen, Carl W.; Hardy, Dwight J.; Swanson, Robert N.; Giardina, William J.; et al.
Journal of Medicinal Chemistry, 1991 , vol. 34, # 1 p. 168 - 174
N-[2-(4-sulphonatephenylamino)-4-methoxy-1,3,5-triazin-6-yl]-4-methylmorpholinium inner salt; sodium hydrogencarbonate in water
5 h; Product distribution / selectivity;
