反应条件
1: N-3-hydroxypropyl-N-methylamine With sodium hydride in dimethyl sulfoxide T=20°C; 1 h; 2: (S)-5-chloro-6-(2,4,6-trifluorophenyl)-N-(1,1,1-trifluoropropan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine in dimethyl sulfoxide T=60°C; 3 h;
参考文献
Zhang, Nan; Ayral-Kaloustian, Semiramis; Nguyen, Thai; Afragola, Jay; Hernandez, Richard; Lucas, Judy; Gibbons, James; Beyer, Carl
Journal of Medicinal Chemistry, 2007 , vol. 50, # 2 p. 319 - 327