1: 100 percent / Et3N; 1percent CuI / 2percent PdCl2(PPh3)2 / 16 h / 60 °C
2: 24 h / 100 °C
3: 41 percent / 10percent CuI / dimethylformamide / 92 h / 100 - 130 °C
View Scheme
参考文献
Zhang, Haiming; Larock, Richard C.
Journal of Organic Chemistry, 2002 , vol. 67, # 20 p. 7048 - 7056