反应条件
1: 1.) NaOEt, 2.) NaI / 1.) EtOH, 0.25 h, 2.) EtOH, RT, 48 h 2: 84 percent / NaN3, NH4Cl / dimethylformamide / 20 h / 105 °C View Scheme
参考文献
Dillard, Robert D.; Carr, F. Patrick; McCullough, Doris; Haisch, Klaus D.; Rinkema, Lynn E.; Fleisch, Jerome H.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 5 p. 911 - 918
