(R)-1-Boc-2-哌嗪甲酸甲酯合成路线 (共 2 条)
反应条件
in methanol; hexane; dichloromethane T=20°C; 16 h;
参考文献
ASTRAZENECA AB; ASTRAZENECA UK LIMITED
Patent: WO2005/26152 A1, 2005 ;
Location in patent: Page/Page column 136 ;
WO 2005/026152 A1
反应条件
lithium aluminium tetrahydride in tetrahydrofuran T=-40 - 20°C; 1 h;
参考文献
ASTRAZENECA AB; ASTRAZENECA UK LIMITED
Patent: WO2005/26152 A1, 2005 ;
Location in patent: Page/Page column 136 ;
WO 2005/026152 A1