反应条件
1: 1.) LDA, 2.) PhN(SO2CF3)2, 3.) Pd(PPh3)4, LiCl, aq. Na2CO3, 4.) H2 / 4.) Pd/C 2: HCl / methanol View Scheme
参考文献
Elliott; Broughton; Cascieri; Chicchi; Huscroft; Kurtz; MacLeod; Sadowski; Stevenson
Bioorganic and Medicinal Chemistry Letters, 1998 , vol. 8, # 14 p. 1851 - 1856