3-三氟甲基苯基溴代乙酰胺合成路线 (共 2 条)
反应条件
in dichloromethane T=10 - 20°C; 1.58333 h;
参考文献
GLAXO GROUP LIMITED; UNIVERSITY OF NOTTINGHAM; BRANCH, Clive, Leslie
Patent: WO2008/92878 A1, 2008 ;
Location in patent: Page/Page column 41-42 ;
WO 2008/092878 A1
反应条件
N-ethyl-N,N-diisopropylamine in dichloromethane T=0°C; 1 h;
参考文献
VERTEX PHARMACEUTICALS INCORPORATED
Patent: WO2005/19190 A2, 2005 ;
Location in patent: Page/Page column 59 ;
WO 2005/019190 A2