反应条件
1: With hydrogenchloride in 1,4-dioxane T=40 - 74°C; 20 h; 2: With sulfuric acid in 1,4-dioxane T=100°C; 7 h;
参考文献
Maerki, H. P.; Binggeli, A.; Bittner, B.; Bohner-Lang, V.; Breu, V.; Bur, D.; Coassolo, Ph.; Clozel, J. P.; D'Arcy, A.; Doebeli, H.; Fischli, W.; et al.
Farmaco, 2001 , vol. 56, # 1-2 p. 21 - 28