反应条件
1: 5-bromopyridin-2-yl amine; 1,1'-carbonothioylbis-1H-imidazole in acetonitrile T=20°C; 15 h; 2: 2-(2-aminoethyl)-thiophene in N,N-dimethyl-formamide T=100°C; 15 h; Further stages.;
参考文献
Uckun, Fatih M.; Tibbles, Heather; Erbeck, Douglas; Venkatachalam, Taracad K.; Qazi, Sanjive
Arzneimittel-Forschung/Drug Research, 2007 , vol. 57, # 4 p. 218 - 226